Experiment 607880

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationMAHON,TM: O'NEILL,LAJ:. (1995). STUDIES INTO THE EFFECT OF THE TYROSINE KINASE INHIBITOR HERBIMYCIN A ON NF-KB ACTIVATION IN T LYMPHOCYTES.. 270(48)
Amount utilized
Compound isolated
DiseaseVS.INTERLEUKIN-1 OR PHORBOL MYRISTATE ACETATE-INDUCED NUCLEAR FACTOR-KAPPA-B STIMULATION. COMPOUND APPEARS TO ACT BY MODIFYING A P50 CYSTEINE RESIDUE THAT PREVENTS ITS BINDING TO NF-KB THEREBY PREVENTING NF-KB'S BINDING TO DNA AND GENE EXPRESSIO ENHANCEMENT.
Dose amount0.2 MICROMOLS
Number1
Qualitative resultACTIVE
AnimalCELL CULTURE
Dose expressionCONC USED