Experiment 623665

Details

PropertyValue
Pharmacology
OrganismCitrus paradisi (RUTACEAE)
CitationHE,K: IYER,KR: HAYES,RN: SINZ,MW: WOOLF,TF: HOLLENBERG,PF:. (1998). INACTIVATION OF CYTOCHROME P450 3A4 BY BERGAMOTTIN, A COMPONENT OF GRAPEFRUIT JUICE.. 11(4)
Amount utilized
Compound isolated
DiseaseMEASURED BY INHIBITION OF LIVER MICROSOMAL ENZYMES INVOLVED IN DEMETHYLATION OF ERYTHROMYCIN AND HYDROXYLATION OF TESTOSTERONE.
Dose amount50.0 MICROMOLS
Number1
Qualitative resultACTIVE
AnimalRAT
Dose expressionCONC USED
ExtractFRUIT JUICE