Experiment 635124

Compounds isolated

Details

PropertyValue
Pharmacology
Administration routeORAL
OrganismEmpty organism
CitationCASTANO,G: MAIS,R: FERNANDEZ,JC: LOPEZ,LE: FERNANDEZ,L:. (1999). A LONG-TERM, OPEN-LABEL STUDY OF THE EFFICACY AND TOLERABILITY OF POLICOSANOL IN PATIENTS WITH HIGH GLOBAL CORONARY RISK.. 60(7)
Amount utilized
Compound isolated
DiseaseA LONG-TERM, OPEN-LABEL STUDY, THE EFFECTS OF POLICOSANOL (20MG/D) WERE INVESTIGATED IN THE TREATMENT OF TYPE II HYPERCHOLESTEROLEMIA IN PATIENTS WITH HIGH GLOBAL CORONARY RISK. AFTER DIETARY STABILIZATION DURING A 5-WEEK BASELINE PERIOD, 68 PATIENTS TOOK POLICOSANOL 20MG ONCE DAILY WITH THE EVENING MEAL FOR 12 MONTHS. AFTER TREATMENT WITH POLICOSANOL, LOW-DENSITY LIPOPROTEIN CHOLESTEROL(LDL-C) AND TOTAL CHOLESTEROL DECREASED SIGNIFICANTLY(P<0.00001) BY 24.7% AND 15.9% RESPECTIVELY, AND HIGH-DENSITY LIPOPROTEIN CHOLESTEROL (HDL-C) INCREASED SIGNIFICANTLY (P<0.0001) BY 31.1%. THE RATIOS OF TOTAL CHOLESTEROL TO HDL-C AND LDL-C DECREASED SIGNIFICANTLY(P<0.00001) BY 29.3% AND 37.8%, RESPECTIVELY. THESE EFFECTS CONTINUED TO TO INCREASE, ALTHOUGH MODERATELY, DURING THE 12-MONTH FOLLOW-UP. AT THE END OF THE STUDY, REDUCTIONS WERE NOTED IN TOTAL CHOLESTEROL(30.0%), LDL-C(44.8%), TOTAL CHOLESTEROL TO HDL-C RATIO(54.1%), AND LDL-C TO HDL-C RATIO(62.7%), WHEREAS HDL-C INCREASED BY 68.5%. TRIGLYCERIDES, WHICH DECREASED SIGNIFICANTLY FROM 4 UNTIL 12 MONTHS, WERE 21.2% LOWER AT 12 MONTHS THAN AT BASELINE. OF 59 PATIENTS WHO COMPLETED THE STUDY, 56(94.4%) HAD REDUCTIONS IN LDL-C >15% AT STUDY COMPLETION. THE TREATMENT WAS WELL TOLERATED; NO DRUG-RELATED CLINICAL OR BIOCHEMICAL ADVERSE EFFECTS(AES) WERE DETECTED. RESULTS OF THE PRESENT STUDY SHOW THAT POLICOSANOL 20MG ONCE DAILY FOR 1 YEAR WAS EFFECTIVE AND WELL TOLERATED IN PATIENTS WITH TYPE II HYPERCHOLESTEROLEMIA AND HIGH GLOBAL CORONARY RISK.
Dose amount20.0 MG
Number3
Qualitative resultACTIVE
AnimalHUMAN ADULT
Per unitDAY
Dose expressionDOSE
GenderGIVEN TO BOTH SEXES