Experiment 635439

Details

PropertyValue
Pharmacology
Administration routeORAL
OrganismEmpty organism
CitationWANG,HL: ZOU,HF: KONG,LA: ZHANG,YK: PANG,HA: SU,CY: LIU,GY: HUI,M: FU,L:. (1999). DETERMINATION OF GINSENOSIDE RG3 IN PLASMA BY SOLID-PHASE EXTRACTION AND HIGH-EPRFORMANCE LIQUID CHROMATOGRAPHY FOR PHARMACOKINETIC STUDY.. 731(2)
Amount utilized
Compound isolated
DiseaseA METHOD USING HIGH-PERFORMANCE LIQUID CHROMATOGRAPHY (HPLC) AND SOLID-PHASE EXTRACTION (SPE) IS DESCRIBED FOR THE DETERMINATION OF GINSENOSIDE RG3 IN HUMAN PLASMA 2.5-ML VOLUME OF PLASMA WAS MIXED WITH 2.5 ML 60% METHANOL AQUEOUS SOLUTION, AND CENTRIFUGED AT 1100 G FOR 10 MIN. THE SEPERNATANT FLUID WAS FURTHER PURIFIED BY SPE WITH 200 MG/5 ML 40 MICRONS OCTADECYL SILICA AND SEPARATION WAS OBTAINED USING A REVERSED-PHASE COLUMN UNDER ISOCRATIC CONDTIONS WITH ULTRAVIOLET ABSORBANCE DETECTION. THE INTRA- AND INTER-DAY PRECISION, DETERMINED AS RELATIVE STANDARD DEVIATIONS, WERE LESS THAN 5.0%, AND METHOD RECOVERY WAS MORE THAN 97%. THE LOWER LIMIT OF QUANTITATION, BASED ON STANDARDS WITH ACCEPTABLE RSDS, WAS 2.5 NG/ML. NO ENDOGENOUS COMPOUNDS WERWE FOUND OT INTERFERE WITH ANALYSIS. A GOOD LINEAR RELATIONSHIP WITH A REGRESSION COEFFICIENT OF 0.9999 IN THE RANGE OF 2.5 TO 200 NG/ML WAS OBSERVED. THIS METHOD HAS BEEN DEMONSTRATED TO BE SUITABLE FOR PHARMACOKINEIC STUDIES IN HUMANS.
Dose amountVAR
Number2
Qualitative resultACTIVE
AnimalHUMAN ADULT
Dose expressionDOSE