Experiment 639010

Details

PropertyValue
Pharmacology
Administration routeORAL
OrganismEmpty organism
CitationINGERSLEV,J: SVENDSEN,TL: MORK,A:. (1997). IS AN EPHEDRINE-CAFFEINE TREATMENT CONTRAINDICATED IN HYPERTENSION?. 21(8)
Amount utilized
Compound isolated
DiseaseA DOUBLE-BLIND, RANDOMIZED, PLACEBO CONTROLLED STUDY OF 5 PARALLEL GROUPS OF OVERWEIGHT PATIENTS FROM GENERAL PRACTICES. 166 PATIENTS WITH BODY MASS INDEX(BMI) < 25 KG/M2 WERE INCLUDED CONSECUTIVELY BY 25 GENERAL PRACTITIONERS IN DENMARK AND RANDOMIZED INTO 5 GROUPS:(1) HYPERTENSIVE PATIENTS TREATED WITH BETA-BLOCKERS AND E+C; (2) HYPERTENSIVE PATIENTS TREATED WITH ANTIHYPERTENSIVE AGENTS OTHER THAN BETA-BLOCKERS, AND E+C; (3) NORMOTENSIVE PATIENTS TREATED WITH E+C; (4) HYPERTENSIVE PATIENTS UNDER ANY ANTIHYPERTENSIVE TREATMENT + PLACEBO; AND (5) NORMOTENSIVE PATIENTS + PLACEBO. ALL PATIENTS WERE INSTRUCTED IN A 1200 KCAL (=5040 KJ) DIET. OF A TOTAL OF 138 PATIENTS AGED 20-74, 112 COMPLETED THE STUDY PROTOCOL, FLUCTUATIONS IN SYSTOLIC + DIASTOLIC BLOOD PRESSURE WERE SEEN IN ALL GROUPS. THE SYSTOLIC BLOOD PRESSURE WAS REDUCED SIGNIFICANTLY (5.5 MM HG) IN THE PATIENTS TREATED WITH ANTIHYPERTENSIVE AGENTS OTHER THAN BETA BLOCKERS, PLUS E+C. IN THE OTHER HYPERTENSIVE GROUPS THE REDUCTION IN BLOOD PRESSURE WAS NOT SIGNIFICANT. IN NORMOTENSIVE PATIENTS TREATED WITH E+C, THE SYSTOLIC AND DIASTOLIC BLOOD PRESSURE DECLINED SIGNIFICANTLY (4.4/3.9 MM HG). AT THE END OF THE TREATMENT PERIOD HEART RATE HAD INCREASED SIGNIFICANTLY (4.9 BEATS/MIN) IN THE GROUP OF NORMOTENSIVE PATIENTS TREATED WITH E+C. BLOOD PRESSURE AND HEART RATE MEASURED BY THE PATIENT AT HOME SHOWED SIMILAR FLUCTUATIONS FROM BASELINE PRIOR TO AND DURING TREATMENT WITH E+C OR PLACEBO. A MEAN LOSS OF WEIGHT OF APPROXIMATELY 4 KG IN 6 WEEKS WAS SIGNIFICANT FOR ALL THE GROUPS. THERE WAS NO SIGNIFICANT DIFFERENCE BETWEEN THE GROUPS DURING THIS SHORT PERIOD OF TREATMENT. IN 56% OF THE PATIENTS TREATED WITH E+C COMPLAINTS/SIDE- EFFECTS RELATED TO MEDICAL TREATMENT WERE FOUND AT QUESTIONING. CORRESPONDING COMPLAINTS OCCURRED IN 21% OF THE PLACEBO TREATED PATIENTS. IN THE E+C TREATED GROUP 7% DROPPED OUT DUE TO SIDE-EFFECTS. IN THE PLACEBO GROUP THERE WERE NO DROPOUTS. CONCLUSIONS: THE STUDY DOES NOT SUPPORT THE ASSUMPTION THAT E+C SHOULD CAUSE A RISE IN BLOOD PRESSURE, ACUTELY OR DURING SHORT TERM TREATMENT IN EITHER NORMOTENSIVE OR HYPERTENSIVE OBESE PATIENTS. THE ANTIHYPERTENSIVE EFFECT OF THE BETA BLOCKERS WAS NOT REVERSED BY E+C. A COMMERCIAL PRODUCT, LETIGEN, WAS USED.
Dose amountVAR
Number1
Qualitative resultINACTIVE
AnimalHUMAN ADULT
Dose expressionDOSE
GenderGIVEN TO BOTH SEXES