Experiment 639073

Worktypes

Details

PropertyValue
Pharmacology
Administration routeORAL
OrganismOenothera biennis (ONAGRACEAE)
CitationPUOLAKKA,J: MAKARAINEN,L: VIINIKKA,L: YLIKORKALA,O:. (1985). BIOCHEMICAL AND CLINICAL EFFECTS OF TREATING THE PREMENSTRUAL SYNDROME WITH PROSTAGLANDIN SYNTHESIS PRECURSORS.. 30(3)
Amount utilized
Compound isolated
DiseaseTHE CLINICAL AND BIOCHEMICAL EFFECTS OF A PROSTAGLANDIN SYNTHESIS PRECURSOR (EFAMOL) CONTAINING LINOLEIC ACID AND ITS METABOLITE, GAMMA-LINOLENIC ACID, WERE STUDIED IN 30 WOMEN WITH SEVERE, INCAPACITATING PREMENSTRUAL SYNDROME. EFAMOL TREATMENT ALLEVIATED THE PREMENSTRUAL SYMPTOMS IN GENERAL AND DEPRESSION ESPECIALLY BETTER THAN DID A PLACEBO. THE CAPACITY OF PLATELETS TO RELEASE THROMBOXANE B2 DURING SPONTANEOUS CLOTTING WAS DECREASED IN PATIENTS UNDERGOING EFAMOL TREATMENT(141+/-59 NG/ML, MEAN +/- SD) AS COMPARED TO THOSE UNDERGOING PLACEBO TREATMENT(186 +/- 44 NG/ML, P<0.01) AND CONTROL SUBJECTS (176 +/-40 NG/ML, N=25, P<0.05. NO CHANGES WERE FOUND IN PLASMA 6-KETO-PROSTAGLANDIN F-1A OR IN FSH,LH, PROLACTIN, PROGESTERONE, ESTRADIOL AND TESTOSTERONE. THE DATA SUGGEST THAT PROSTAGLANDINS MIGHT PLAY A ROLE IN THE PATHOPHYSIOLOGY OF THE PREMENSTRUAL SYNDROME. A COMMERCIAL PRODUCT, EFAMOL, WAS USED.
Dose amount3.0 GM
Number1
Qualitative resultACTIVE
AnimalHUMAN ADULT
Per unitDAY
Dose expressionDOSE
ExtractSEED OIL
GenderFEMALE