Experiment 642112

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationRAO,KN: VENKATACHALAM,SR:. (1999). DIHYDROFOLATE REDUCTASE AND CELL GROWTH ACTIVITY INHIBITION BY THE BETA-CARBOLINE-BENZOQUINOLIZIDINE PLANT ALKALOID DEOXYTUBULOSINE FROM ALANGIUM LAMARCKII: ITS POTENTIAL AS AN ANTIMICROBIAL AND ANTICANCER AGENT.. 7(6)
Amount utilized
Compound isolated
DiseaseINHIBITS L. LEICHMANNI'S DHFR ACTIVITY AT AN IC50 VALUE OF 30NM. > 75 MM RESULTS IN COMPLETE LOSS OF ENZYME ACTIVITY SUGGESTING IT TO HAVE A HIGH POTENTIAL AS AN ANTITUMOR AGENT.
Dose amount30.0 MICROMOLS
Number1
Qualitative resultACTIVE
AnimalCELL CULTURE
Per unitML
Dose expressionIC50