Experiment 642179

Compounds isolated

Details

PropertyValue
Pharmacology
Administration routeORAL
OrganismEmpty organism
CitationZUTSHI,RK: SINGH,R: ZUTSHI,U: JOHRI,RK: ATAL,CK:. (1985). INFLUENCE OF PIPERINE ON RIFAMPICIN BLOOD LEVELS IN PATIENTS OF PULMONARY TUBERCULOSIS.. 33(3)
Amount utilized
Compound isolated
DiseaseTHE INFLUENCE OF PIPERINE ON RIFAMPICIN LEVELS IN 14 PATIENTS(7 MALES, 7 FEMALES) OF PULMONARY TUBERCULOSIS WAS STUDIED. THE PATIENTS WERE FED 450 MG RIFAMPICIN AND BLOOD LEVELS OF THE DRUG DETERMINED BY UV SPECTROPHOTOMETER O.25, 0.5, 1,2,4,8 AND 12 HOURS LATER. AFTER FIVE DAYS RIFAMPICIN (450 MG) WAS COADMINISTERED WITH PIPERINE (50 MG) AND THE BLOOD LEVELS OF RIFAMPICIN WERE AGAIN MONITORED. A HIGHLY SIGNIFICANT(P< 0.01) INCREASE IN RIFAMPICIN PLASMA LEVELS AND AREA UNDER THE DRUG CONCENTRATION VERSUS TIME CURVE WAS NOTICED IN BOTH THE SEXES WHEN PIPERINE WAS COADMINISTERED, ALTHOUGH THERE WAS VARIATION IN THE T MAX. THE SEX DEPENDENT DIFFERENCE OBSERVED WAS STATISTICALLY INSIGNIFICANT.
Dose amount50.0 MG
Number1
Qualitative resultACTIVE
AnimalHUMAN ADULT
Per unitDAY
Dose expressionDOSE
GenderGIVEN TO BOTH SEXES