Experiment 642206

Compounds isolated

Details

PropertyValue
Pharmacology
Administration routeORAL
OrganismEmpty organism
CitationHOLODNIV,M: KOCH,J: MISTAL,M: SCHMIDT,JM: KHANDWALA,A: PENNINGTON,JE: PORTER,SB:. (1999). A DOUBLE BLIND, RANDOMIZED, PLACEBO-CONTROLLED PHASE II STUDY TO ASSESS THE SAFETY AND EFICACY OF ORALLY ADMINISTERED SP-303 FOR THE SYMPTOMATIC TREATED OF DIARRHEA IN PATIENTS WITH AIDS.. 94(11)
Amount utilized
Compound isolated
DiseaseMULTICENTER PHASE II RANDOMIZED DOUBLE BLIND PLACEBO-CONTROLLED STUDY. HIV-POSITIVE SUBJECTS AND AIDS-DEFINING ILLNESS WERE ADMITTED TO AN INPATIENT STUDY UNIT. SUBJECTS RECIEVED 500 MG OF SP-303 OR PLACEBO EVERY 6 HOUR FOR 96 HOURS. STOOL FREQUENCY AND WEIGHTS WERE RECORDED. DAILY MEASURES ANALYSIS OVER 4 DAYS OF TREATMENT DEMONSTRATED THAT SP-303 SUBJECTS HAD A SIGNIFICANT REDUCTION IN STOOL WEIGHT AND ABNORMAL STOOL FREQUENCY WHEN COMPARED TO PLACEBO TREATED SUBJECTS. SP-303 IS SAFE AND WELL TOLERATED. SP-303 IS EFFECTIVE IN REDUCING STOOL WEIGHT AND FREQUENCY IN PATIENTS WITH AIDS AND DIARRHEA.
Dose amount2.0 GM
Number1
Qualitative resultACTIVE
AnimalHUMAN ADULT
Per unitDAY
Dose expressionDOSE
GenderGIVEN TO BOTH SEXES