Experiment 646370
Worktypes
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | ORAL |
| Organism | Citrus paradisi (RUTACEAE) |
| Citation | ZAIDENSTEIN,R: DISHI,V: GIPS,M: SOBACK,S: COHEN,N: WEISSGARTEN,J: BLATT,A: GOLIK,A:. (1998). THE EFFECT OF GRAPEFRUIT JUICE ON THE PHARMACOKINETICS OF ORALLY ADMINISTERED VERAPAMIL.. 54(4) |
| Amount utilized | |
| Compound isolated | |
| Disease | AUC(VERAPAMIL)/AUC(METABOLITE D-617) WAS SLIGHTLY BUT SIGNIFICANTLY INCREASED. C MAX, T MAX, AUC(VERAPAMIL) AND AUC(METABOLITE D-617) NOT AFFECTED BY GRAPEFRUIT JUICE. STUDY WAS CONDUCTED ON HYPERTENSIVE PATIENTS. |
| Dose amount | 200.0 ML |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | HUMAN ADULT |
| Per unit | DAY |
| Dose expression | DOSE |
| Extract | FRUIT JUICE |