Experiment 647113
Worktypes
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | ORAL |
| Organism | Citrus paradisi (RUTACEAE) |
| Citation | JOSEFESSON,M: JACKRISSON,AL: AHLNER,J:. (1996). EFFECT OF GRAPEFRUIT JUICE ON THE PHARMACOKINETICS OF AMLODIPINE IN HEALTHY VOLUNTEERS.. 51(2) |
| Amount utilized | |
| Compound isolated | |
| Disease | A RANDOMIZED OPEN CROSSOVER STUDY DESIGN COMPARED THE EFFECT OF A SINGLE DOSE OF AMLODIPINE TAKEN WITH GRAPEFRUIT JUICE VS. WATER. CMAX WAS 115% AND AUC(0.72H) WAS 116% COMPARED WITH WATER BUT TMAX WAS NOT SIGNIFICANTLY CHANGED. |
| Dose amount | 250.0 ML |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | HUMAN ADULT |
| Per unit | DAY |
| Dose expression | DOSE |
| Extract | FRUIT JUICE |
| Gender | MALE |