Experiment 647134
Worktypes
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | ORAL |
| Organism | Citrus paradisi (RUTACEAE) |
| Citation | TAKANAGA,H: OHNISHI,A: MATSUO,H: MURAKAMI,H: SATA,H: KURODA,K: URAE,A: HIGUCHI,S: SAWADA,Y:. (2000). PHARMACOKINETIC ANALYSIS OF FELODIPINE-GRAPEFRUIT JUICE INTERACTION BASED ON AN IRREVERSIBLE ENZYME INHIBITION MODEL.. 49(1) |
| Amount utilized | |
| Compound isolated | |
| Disease | FELODIPINE AS A MODEL DRUG CONSTRUCTED A PHARMACOKINETIC MODEL BASED ON IRREVERSIBLE INHIBITION OF INTESTINAL CYTOCHROME P450 3A4 BY GRAPEFRUIT JUICE(GFJ). GFJ-FELODIPINE INTERACTION INCREASES WITH INCREASING FREQUENCY AND AMOUNT OF GFJ INGESTION. |
| Dose amount | VAR |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | HUMAN ADULT |
| Dose expression | DOSE |
| Extract | FRUIT JUICE |
| Gender | GIVEN TO BOTH SEXES |