Experiment 652674

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationVANSAL,SS: FELLER,DR:. (1999). DIRECT EFFECTS OF EPHEDRINE ISOMERS ON HUMAN BETA-ADRENERGIC RECEPTOR SUBTYPES.. 58(5)
Amount utilized
Compound isolated
DiseaseON HUMAN B-ADRENERGIC(B1-AR) IT WAS SHOWN THAT ONLY 1R,2S-EPHEDRINE SHOWED SIGNIFICANT AGONIST ACTIVITY ON HUMAN B3-AR WITH AN EC50=45 MM AND A MAXIMAL RESPONSE OF 31%. AND IT HAS WEAK PARTIAL AGONIST ACTIVITY ON B3-AR.
Dose amount45.0 MICROMOLS
Number1
Qualitative resultACTIVE
AnimalCELL CULTURE
Per unitSQ M BODY SURFACE
Dose expressionED50