Experiment 652677
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Empty organism |
| Citation | VANSAL,SS: FELLER,DR:. (1999). DIRECT EFFECTS OF EPHEDRINE ISOMERS ON HUMAN BETA-ADRENERGIC RECEPTOR SUBTYPES.. 58(5) |
| Amount utilized | |
| Compound isolated | |
| Disease | ON HUMAN B-ADRENERGIC(B1-AR) IT WAS SHOWN THAT ONLY 1R,2S-EPHEDRINE SHOWED SIGNIFICANT AGONIST ACTIVITY ON HUMAN B3-AR WITH AN EC50=45 MM AND A MAXIMAL RESPONSE OF 31%. AND IT HAS WEAK PARTIAL AGONIST ACTIVITY ON B3-AR. |
| Dose amount | 309.0 MICROMOLS |
| Number | 4 |
| Qualitative result | INACTIVE |
| Animal | CELL CULTURE |
| Dose expression | ED50 |