Experiment 66665
Worktypes
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | ORAL |
| Organism | Aesculus hippocastanum (HIPPOCASTANACEAE) |
| Citation | OSCHMANN,R: BIBER,A: LANG,F: STUMPF,H: KUNZ,K:. (1996). PHARMACOKINETICS OF BETA-ESCIN AFTER ADMINISTRATION OF DIFFERENT AESCULUS-EXTRACT CONTAINING FORMULATIONS.. 51(8) |
| Amount utilized | |
| Compound isolated | |
| Disease | WITH A SPECIFIC RADIOIMMUNOASSAY THE PHARMACOKINETICS AND RELATIVE BIOAVAILABILITY OF ESCIN WAS MEASURED AFTER ADMINISTRATION OF DIFFERENT FORMULATIONS CONTAINING ASECULUS-EXTRACT. OF SPECIAL INTEREST WAS THE RELATIVE BIOAVAILABILITY OF ESCIN AFTER ADMINISTRATION OF A NEWLY DEVELOPED FILMCOATED TABLET WITH SUSTAINED RELEASE IN COMPARISON TO A REFERENCE FORMULATION. IN A CROSS-OVER STEADY-STATE STUDY IN 24 VOLUNTEERS BIOEQUIVALENCE OF TEST AND REFERENCE PREPARATION COULD BE DEMONSTRATED. THE 90% CONFIDENCE INTERVAL OF THE AUC(O-TAU) WAS 98.3 TO 120.9%. |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | HUMAN ADULT |
| Dose expression | DOSE |
| Extract | SAPONIN FRACTION |
| Gender | GIVEN TO BOTH SEXES |