Experiment 67452
Worktypes
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | ORAL |
| Organism | Citrus paradisi (RUTACEAE) |
| Citation | BISTRUP,C: NIELSEN,FT: JEPPESEN,UE: DIEPERINK,H:. (2001). EFFECT OF GRAPEFRUIT JUICE OF SANDIMMUN NEORAL ABSORPTION AMONG STABLE RENAL ALLOGRAFT RECIPIENTS.. 16(2) |
| Amount utilized | |
| Compound isolated | |
| Disease | A RANDOMIZED CROSS-OVER STUDY INVOLVING 8 STABLE RENAL TRANSPLANT PATIENTS. IN TWO 8-HR STUDY PERIODS WITH A 4-WK INTERVAL THE EFFECT OF GRAPEFRUIT JUICE INGESTION ON CYCLOSPORIN A LEVELS WAS ASSESSED. THE MEDIAN AREA-UNDER-THE-CURVE WAS INCREASED BY 38% FOLLOWING CO-ADMINISTRATION. NO CHANGES IN C-MAX, T-MAX, OR T1/2. |
| Dose amount | 500.0 ML |
| Number | 2 |
| Qualitative result | ACTIVE |
| Animal | HUMAN ADULT |
| Per unit | DAY |
| Dose expression | DOSE |
| Extract | JUICE |
| Gender | GIVEN TO BOTH SEXES |