Experiment 67591
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | ORAL |
| Organism | Empty organism |
| Citation | BACHUS,R: BICKEL,U: THOMSEN,T: ROOTS,I: KEWITZ,H:. (1999). THE O-DEMETHYLATION OF THE ANTIDEMENTIA DRUG GALANTHAMINE IS CATALYSED BY CYTOCHROME P450 2D6.. 9(6) |
| Amount utilized | |
| Compound isolated | |
| Disease | VS.EIGHT YOUNG MEN; METABOLIZED TO O-DEMETHYLGALANTHAMINE WITH VMAX 5.2 NMOL/MG PROTEIN/H AND KM 187 MICRO MOLAR. |
| Dose amount | 10.0 MG |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | HUMAN ADULT |
| Dose expression | DOSE |
| Gender | MALE |