Experiment 67641

Compounds isolated

Details

PropertyValue
Pharmacology
Administration routeORAL
OrganismEmpty organism
CitationKAMIMORI,GH: HEADLEY,DB: THORNE,DR: OTTERSTETTER,DR: BELENKY,G:. (2000). EFFECT OF THREE CAFFEINE DOSES ON PLASMA CATECHOLAMINES AND ALERTNESS DURING PROLONGED WAKEFULNESS.. 56(8)
Amount utilized
Compound isolated
DiseaseFOLLOWING 49H OF PROLONGED WAKEFULNESS, EACH OF 50 HEALTHY MALES ORALLY INGESTED EITHER A PLACEBO OR ONE OF THREE DOSES OF CAFFEINE, 2.1 (LOW), 4.3(MEDIUM), OR 8.6 MG KG-1 BODY WEIGHT (HIGH), IN A RANDOMIZED DOUBLE-BLIND DESIGN. WAKEFULNESS CONTINUED FOR AN ADDITIONAL 12H DURING WHICH VENOUS BLOOD SAMPLES WERE COLLECTED FOR CATECHOLAMINE AND CAFFEINE ANALYSIS. A SLEEP LATENCY TEST, THE STANFORD SLEEPINESS SCALE, AND A CHOICE REACTION TIME TEST WERE ADMINISTERED AS MEASURES OF ALERTNESS. CAFFEINE HAD NO SIGNIFICANT EFFECT ON NORADRENALINE, BUT ADRENALINE WAS SIGNIFICANTLY INCREASED BETWEEN 1H AND 4H POST-DOSING IN THE HIGH DOSE GROUP COMPARED WITH A PLACEBO GROUP. FOLLOWING CAFFEINE ADMINISTRATION, RESPONSES TO SLEEP LATENCY, SLEEPINESS SCORES, AND REACTION TIME SCORES SHOWED DOSE-RELATED CHANGES THAT WERE EXHIBITED BY SIGNIFICANT CORRELATION COEFFICIENTS.
Dose amountVAR
Number1
Qualitative resultACTIVE
AnimalHUMAN ADULT
Dose expressionDOSE
GenderMALE