Experiment 676831
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Spachea correae (MALPIGHIACEAE) |
| Citation | FELIX,JP: BUGIANESI,RM: SCHMALHOFER,WA: BORRIS,R: GOETZ,MA: HENSENS,OD: BAO,JM: KAYSER,F: PARSONS,WH: RUPPRECHT,K: GARCIA,ML: KACZOROWSKI,GJ: SLAUGHTER,RS:. (1999). IDENTIFICATION AND BIOCHEMICAL CHARACTERIZATION OF A NOVEL NORTRITERPENE INHIBITOR OF THE HUMAN LYMPHOCYTE VOLTAGE-GATED POTASSIUM CHANNEL, KV1.3.. 38(16) |
| Amount utilized | |
| Compound isolated | |
| Disease | POTENCY OF INHIBITION OF 86RB+ EFFLUX FROM CHO/KV1.3 CELLS INCREASE WITH TIME OF PREINCUBATION. |
| Dose amount | 12.0 NANOMOLS |
| Number | 5 |
| Qualitative result | ACTIVE |
| Animal | CELL CULTURE |
| Dose expression | IC50 |