Experiment 677897

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationLYB,G: KNORRE,A: SCHMIDT,TJ: PAHL,HL: MERFORT,I:. (1998). THE ANTI-INFLAMMATORY SESQUITERPENE LACTONE HELENALIN INHIBITS THE TRANSCRIPTION FACTOR NF-KB BY DIRECTLY TARGETING P65.. 273(50)
Amount utilized
Compound isolated
DiseaseTHESE DATE SHOW THAT NITHER IKAPABET ADEGRADATION NOR NF-KAPABETA NUCLEAR TRANSLOCAITON ARE INHIBITED, HELENAL SELECTIVELY ALKYLATES THE P65 SUBUNIT OF NF-KAPABETA.
Dose amountVAR
Number1
Qualitative resultACTIVE
AnimalCELL CULTURE
Dose expressionCONC USED