Experiment 67837

Compounds isolated

Details

PropertyValue
Pharmacology
Administration routeIV
OrganismEmpty organism
CitationBLACKHALL,FH: RANSON,M: RADFORD,JA: HACOCK,BW: SOUKOP,M: MC GOWN,AT: ROBBINS,A: HALBERT,G: JAYSON,GC:. (2001). A PHASE II TRIAL OF BRYOSTATIN 1 IN PATIENTS WITH NON-HODGKIN'S LYMPHOMA.. 84(4)
Amount utilized
Compound isolated
DiseaseIN THIS PHASE II STUDY, 17 PATIENTS WITH PROGRESSIVE NON-HODGKIN'S LYMPHOMA PREVIOUSLY TREATED WITH CHEMOTHERAPHY, RECEIVED A MEDIAN OF 6 (RANGE 1-9) INTRAVENOUS INFUSIONS OF 25 UG/M2 BRYOSTATIN 1 GIVEN ONCE WEEKLY OVER 24 HOURS. IN 14 EVALUABLE PATIENTS NO RESPONSES WERE SEEN. STABLE DISEASE WAS ATTAINED IN ONE PATIENT FOR 9 MONTHS. THE PRINCIPAL TOXICITIES WERE MYALGIA AND PHLEBITIS.
Dose amount25.0 MCG
Number1
Qualitative resultINACTIVE
AnimalHUMAN ADULT
Per unitSQ M BODY SURFACE
Dose expressionDOSE
GenderGIVEN TO BOTH SEXES