Experiment 68063

Worktypes

Details

PropertyValue
Pharmacology
Administration routeORAL
OrganismTrifolium pratense (FABACEAE)
CitationHALE,GE: HUGHES,CL: ROBBOY,SJ: AGARWAL,SK: BIEVRE,M:. (2001). A DOUBLE-BLIND RANDOMIZED STUDY ON THE EFFECTS OF RED CLOVER ISOFLAVONES ON THE ENDOMETRIUM.. 8(5)
Amount utilized
Compound isolated
DiseaseIN A DOUBLE-BLIND, RANDOMIZED, CONTROLLED STUDY, 30 WOMEN BETWEEN THE AGES OF 45 AND 50 YEARS CONSENTED TO AN ENDOMETRIAL BIOPSY BEFORE AND AFTER A 3-MONTH COURSE OF EITHER PLACEBO OR ACTIVE ISOFLAVONE EXTRACT. THE BIOPSIES WERE TIMED AS CLOSE AS POSSIBLE TO DAYS 7-11 OF THE MENSTRUAL CYCLE, AND SIMULTANEOUS MEASUREMENTS OF TRANSVAGINAL ENDOMETRIAL THICKNESS, UTERINE ARTERY DOPPLER, HORMONE PROFILES, LIPIDS, AND BONE MARKERS WERE PERFORMED.OF 30 WOMEN, 2 DID NOT RETURN FOR A SECOND BIOPSY, AND A THIRD HAD AN UNSUCCESSFUL SECOND BIOPSY. FOUR SUBJECTS WERE EXCLUDED FROM THE INTENTION TO TREAT ANALYSIS BECAUSE THEY DID NOT HAVE A MENSTRUAL BLEED WITHIN THE TIME FRAME OF THE STUDY (3 SUBJECTS) OR WERE TESTED ON DAY 13 INSTEAD OF BETWEEN DAYS 7 AND 11 OF THE CYCLE (1 SUBJECT).THERE WAS NO CHANGE IN THE KI-67 PROLIFERATION INDEX AFTER TREATMENT IN EITHER GROUP. EIGHT SUBJECTS IN THE PLACEBO GROUP AND EIGHT IN THE P-07 GROUP HAD PROLIFERATIVE ENDOMETRIAL BIOPSIES THAT WERE SYNCHRONIZED WITH ESTRADIOL LEVELS AT BASELINE AND POST-TREATMENT, AND ANALYSIS OF THESE SUBJECTS REVEALED NO DETECTABLE CHANGE IN THE RELATIONSHIP BETWEEN ESTRADIOL LEVELS AND KI-67 WITH TREATMENT IN EITHER GROUP. THERE WAS NO CHANGE IN FASTING LIPIDS, BONE MARKERS, UTERINE DOPPLER RESISTANCE, OR PULSATILITY INDEX.
Dose amount50.0 MG
Number1
Qualitative resultINACTIVE
AnimalHUMAN ADULT
Dose expressionDOSE
ExtractFLAVONOID FRACTION
GenderFEMALE