Experiment 68635

Details

PropertyValue
Administration routeORAL
OrganismCitrus paradisi (RUTACEAE)
CitationOZDEMIR,V: KALOW,W: OKEY,AB: LAM,MSM: ALBERS,LJ: REIST,C: FOURIE,J:. (2001). TREATMENT-RESISTANCE TO CLOZAPINE IN ASSOCIATION WITH ULTRARAPID CYP1A2 ACTIVITY AND THE C->A POLYMORPHISM IN INTRON 1 OF THE CYP1A2 GENE: EFFECT OF GRAPEFRUIT JUICE AND LOW-DOSE FLUVOXAMINE.. 21(6)
Amount utilized
Compound isolated
DiseaseCO-ADMINISTRATION OF CLOZAPINE(750 MG 3TIMES DAILY) WITH GRAPEFRUIT JUICE DID NOT PRODUCE ANY CHANGE IN CLOZAPINE CONCENTRATIONS OR SEVERITY OF PSYCHOSID.
Dose amount375.0 ML
Number1
Qualitative resultINACTIVE
AnimalHUMAN ADULT
Per unitDAY
Dose expressionDOSE
ExtractFRUIT JUICE
GenderMALE