Experiment 68659

Compounds isolated

Details

PropertyValue
Pharmacology
Administration routeIV
OrganismEmpty organism
CitationBHARGAVA,P: MARSHALL,JL: DAHUT,W: RIZVI,N: TROCKY,N: WILLIAMS,JI: HAIT,H: SONG,S: HOLROYD,KJ: HAWKINS,MJ:. (2001). A PHASE I AND PHARMACOKINETIC STUDY OF SQUALAMINE, A NOVEL ANTIANGIOGENIC AGENT, IN PATIENTS WITH ADVANCED CANCERS.. 7(12)
Amount utilized
Compound isolated
DiseaseA PHASE I AND PHARMACOKINETIC STUDY OF SQUALAMINE, A NOVEL ANTIANGIOGENIC AGENT IN ADVANCED CANCER PATIENTS, SHOWED THE BEST TOLERATED DOSE RATE AT 120H CONTINOUS INFUSION (1V) 192MG PER M-2 PER DAY BUT PATIENTS WITHOUT PRIOR EXPOSURE TO SQUALAMINE APPEARED TO TOLERATE A DOSE RATE OF 384,H/M-2/DAY WITHOUT DLT.
Dose amount192.0 MG
Number1
Qualitative resultACTIVE
AnimalHUMAN ADULT
Per unitDAY
Dose expressionDOSE
GenderGIVEN TO BOTH SEXES