Experiment 68996

Worktypes

Details

PropertyValue
Pharmacology
Administration routeORAL
OrganismSerenoa repens (ARECACEAE)
CitationDEBRUYNE,F: KOCH,G: BOYLE,P: CALAIS DA SILVA,F: GILLENWATER,JG: HAMDY,FC: PERRIN,P: TEILLAC,P: VELA NAVARRETE,R: RAYNAUD,JP:. (2002). COMPARISON OF A PHYTOTHERAPEUTIC AGENT (PERMIXON) WITH AN BETA-BLOCKER (TAMSULOSIN) IN THE TREATMENT OF BENIGN PROSTATIC HYPERPLASIA: A 1-YEAR RANDOMIZED INTERNATIONAL STUDY.. 41(5)
Amount utilized
Compound isolated
DiseaseLIPIDO-STEROLIC EXT. OF SERENOA REPENS (LSESR)-PERMIXON-HAS BEEN SHOWN TO HAVE AN EQUIV. EFFICACY TO FINASTERIDE IN PATIENTS WITH BENIGN PROSTATIC HYPERPLASIA (BPH), TO DATE, THERE HAS BEEN NO VALID COMPARISON OF PHYTOTHERAPY WITH ALPHA- BLOCKERS. THE AIM OF THIS STUDY WAS TO ASSESS THE EQUIV. EFFICACY OF PERMIXON AND TAMSULOSIN. EIGHT HUNDRED AND ELEVEN MEN WITH SYMPTOMATIC BPH (I-PSS>10) WERE RECRUITED IN 11 EUROPEAN COUNTRIES FOR A 12-MO, DOUBLE-BLIND RANDOMIZED TRIAL. AFTER A 4-WK RUN-IN PERIOD, 704 PATIENTS WERE RANDOMLY ASSIGNED TO EITHER TAMSULOSIN O.4 MG/DAY(N=345) OR PERMIXON 320 MG/DAY (N=350). I-PSS, QOL AND Q-MAX WERE EVALUATED AT BASELINE AND PERIODICALLY FOR 1 YR. PROSTATE VOL. AND SERUM PROSTATE- SPECIFIC ANTIGEN (PSA) WERE MEASURED AT SELECTION AND AT ENDPOINT. THE ENDPOINT ANAL. WAS PERFORMED ON THE PER-PROTOCOL POPULATION OF 542 PATIENTS (TAMSULOSIN: N=273; PERMIXON: N=269). AT 12 MO, I-PSS DECREASED BY 4.4 IN EACH GROUP AND NO DIFFERENCES WERE OBSD. IN EITHER IRRITATIVE OR OBSTRUCTIVE SYMPTOM IMPROVEMENTS. THE INCREASE IN Q-MAX WAS SIMILAR IN BOTH TREATMENT GROUPS (1.8ML/S PERMIXON, 1.9 ML/S TAMSULOSIN). PSA REMAINED STABLE WHILE PROSTATE VOL. DECREASED SLIGHTLY IN THE PERMIXON-TREATED PATIENTS. THE TWO COMPDS. WERE WELL TOLERATED, HOWEVER, EJACULATION DISORDERS OCCURRED MORE FREQUENTLY IN THE TAMSULOSIN GROUP. THIS STUDY DEMONSTRATES THAT PERMIXON AND TAMSULOSIN ARE EQUIV. IN THE MEDICAL TREATMENT OF LOWER URINARY TRACT SYMPTOMS IN MEN WITH BPH, DURING AND UP TO 12 MO OF THERAPY.
Dose amount320.0 MG
Number2
Qualitative resultINACTIVE
AnimalHUMAN ADULT
Per unitDAY
Dose expressionDOSE
ExtractFIXED OIL
GenderMALE