Experiment 69473
Worktypes
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | ORAL |
| Organism | Citrus paradisi (RUTACEAE) |
| Citation | CASTRO,N: JUNG,H: MEDINEA,R: GONZALEZ-ESQUIVEL,D: LOPEZ,M: SOTELO,J:. (2002). INTERACTION BETWEEN GRAPEFRUIT JUICE AND PRAZIQUANTEL IN HUMANS.. 46(5) |
| Amount utilized | |
| Compound isolated | |
| Disease | +128.5 NG/ML; AND CMAX FOR GRAPEFRUIT JUICE TREATMENT, 1,037.65+205.7 NG/ML, P<0.05). NO STATISTICALLY SIGNIFICANT DIFFERENCES WERE FOUND IN THE TIME TO MAXIMUM CONCENTRATION OF DRUG IN PLASMA OR ELIMINATION HALF-TIME. AFTER A SINGLE ORAL DOSE PF PRAZIQUANTEL WITH 250 ML OF GRAPEFRUIT JUICE, THE AREA UNDER THE CONCENTRATION-TIME CURVE AND THE MAXIMUM CONCENTRATION IN PLASMA OF PRAZIQUANTEL (CMAX) WERE SIGNIFICANTLY INCREASED (CMAX FOR WATER TREATMENT, 637.71 |
| Dose amount | 250.0 ML |
| Number | 1 |
| Qualitative result | INACTIVE |
| Animal | HUMAN ADULT |
| Dose expression | DOSE |
| Extract | JUICE |
| Gender | GIVEN TO BOTH SEXES |