Experiment 69484

Worktypes

Details

PropertyValue
Pharmacology
Administration routeORAL
OrganismCamellia sinensis (THEACEAE)
CitationJATOI,A: ELLISON,N: BURCH,PA: SLOAN,JA: DAKHIL,SR: NOVOTNY,P: TAN,W: FITCH,TR: ROWLAND,KM: YOUNG,CYF: FLYNN,PJ:. (2003). A PHASE II TRIAL OF GREEN TEA IN THE TREATMENT OF PATIENTS WITH ANDROGEN INDEPENDENT METASTATIC PROSTATE CARCINOMA.. 97(6)
Amount utilized
Compound isolated
DiseasePHASE II TRIAL TO EXPLORE GREEN TEA'S ANTINEOPLASTIC EFFECTS IN PATIENTS WITH ANDROGEN-INDEPENDENT PROSTATE CARCINOMA. STUDY EVALUATED 42 PATIENTS WHO WERE ASYMPTOMATIC AND HAD MANIFESTED, PROGRESSIVE PROSTATE SPECIFIC ANTIGEN (PSA) ELEVATION WITH HORMONE THERAPY. CONTINUED USE OF LUTEINIZING HORMONE-RELEASING HORMONE AGONIST WAS PERMITTED; HOWEVER, PATIENTS WERE INELIGIBLE IF THEY HAD RECEIVED OTHER TREATMENTS FOR THEIR DISEASE IN THE PRECEDING 4 WEEKS OR IF THEY HAD RECEIVED A LONG-ACTING ANTIANDROGEN THERAPY IN THE PRECEDING 6 WEEKS. PATIENTS WERE INSTRUCTED TO TAKE 6 GRAMS OF GREEN TEA PER DAY ORALLY IN 6 DIVIDED DOSES. EACH DOSE CONTAINED 100 CALORIES AND 46 MG OF CAFFEINE. PATIENTS WERE MONITORED MONTHLY FOR RESPONSE AND TOXICITY. TUMOR RESPONSE, DEFINED AS A DECLINE >/= 50% IN THE BASELINE PSA VALUE, OCCURRED IN A SINGLE PATIENT, OR 2% OF THE COHORT (95% CONFIDENCE INTERVAL, 1-14%). THIS ONE RESPONSE WAS NOT SUSTAINED BEYOND 2 MONTHS. AT THE END OF THE FIRST MONTH, THE MEDIAN CHANGE IN THE PSA VALUE FROM BASELINE FOR THE COHORT INCREASED BY 43%. GREEN TEA TOXICITY, USUALLY GRADE 1 OR 2, OCCURRED IN 69% OF PATIENTS AND INCLUDED NAUSEA, EMESIS, INSOMNIA, FATIGUE, DIARRHEA, ABDOMINAL PAIN, AND CONFUSION. HOWEVER, SIX EPISODES OF GRADE 3 TOXICITY AND ONE EPISODE OF GRADE 4 TOXICITY ALSO OCCURRED, WITH THE LATTER MANIFESTING AS SEVERE CONFUSION. CONCLUSIONS: GREEN TEA CARRIES LIMITED ANTINEOPLASTIC ACTIVITY, AS DEFINED BY A DECLINE IN PSA LEVELS, AMONG PATIENTS WITH ANDROGEN INDEPENDENT PROSTATE CARCINOMA.
Dose amount36.0 GM
Number1
Qualitative resultINACTIVE
AnimalHUMAN ADULT
Per unitDAY
Dose expressionDOSE
ExtractH2O EXT
GenderMALE