Experiment 73268
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | ORAL |
| Organism | Empty organism |
| Citation | DE SANTANA,CF: LINS,LJP: ASFORA,JJ: MELO,AM: GONCALVES,O: DELIMA: D'ALBUQUERQUE,IL:. (1981). PRIMARY OBSERVATIONS OF THE USE OF LAPACHOL IN HUMAN CARRIERS OF MALIGNANT NEOPLASMS.. 20(1/2) |
| Amount utilized | |
| Compound isolated | |
| Disease | NINE PATIENTS WITH MALIGNANT CARCINOMA WERE TREATED DAILY FOR 30 TO AS LONG AS 720 DAYS. PARTIAL OBJECTIVE RESPONSE WAS SEEN IN 2 PATIENTS WITH LESION REDUCTION OF 20-30%. ALL PATIENTS EXPERIENCED A REDUCTION OF PAIN. TOXICITY CONSISTED MAINLY OF NAUSEA AND VOMITING, WITH RARE DIARRHEA. NO HEMATOLOGICAL TOXICITY WAS DETECTED AND THERE WERE NO UNUSUAL RESULTS IN URINARY ANALYSIS. |
| Dose amount | 20-30 MG |
| Number | 1 |
| Qualitative result | EQUIVOCAL |
| Animal | HUMAN ADULT |
| Per unit | KG |
| Dose expression | DOSE |