Experiment 755716
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Empty organism |
| Citation | ASANO,T: KUSHIDA,H: SADAKANE,C: ISHIHARA,K: WAKUI,Y: YANAGISAWA,T: KIMURA,M: KAMEI,H: YOSHIDA,T:. (2001). METABOLISM OF IPECAC ALKALOIDS CEPHAELINE AND EMETINE BY HUMAN HEPATIC MICROSOMAL CYTOCHROME P450S, AND THEIR INHIBITORY EFFECTS ON P450 ENZYME ACTIVITIES.. 24(6) |
| Amount utilized | |
| Compound isolated | |
| Disease | VS.CYP2D6 AND CYP3A4 SUBSTRATE. |
| Dose amount | 80.0 MICROMOLS |
| Number | 3 |
| Qualitative result | ACTIVE |
| Animal | HUMAN ADULT |
| Dose expression | IC50 |