Experiment 759056
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Empty organism |
| Citation | ELTZE,M: GREBE,T: MICHEL,MC: CZYBORRA,P: ULLRICH,B:. (2002). AFFINITY PROFILE AT ALPHA-1- AND ALPHA-2-ADRENOCEPTOR SUBTYPES AND IN VITRO CARDIOVASCULAR ACTIONS OF (+)-BOLDINE.. 443(1/3) |
| Amount utilized | |
| Compound isolated | |
| Disease | THESE DATA REVEAL THAT (+)-BOLDINE, EXCEPT FOR ITS MODERATE SELECTIVITY (15 TO 25-FOLD) FOR ALPHA1A-ADRENOCEPTORS, DOES NOT DISCRIMINATE BETWEEN THE ALPHA1-ADRENOCEPTOR SUBTYPES B AND D AND ALPHA2-ADRENOCEPTOR SUBTYPES A, B AND C, AT WHICH THE DRUG CONSISITENTLY DISPLAYS MICROMOLAR AFFINITY. |
| Dose amount | VAR |
| Number | 1 |
| Qualitative result | ACTIVE |
| Dose expression | CONC USED |