Experiment 75980
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | IV |
| Organism | Empty organism |
| Citation | DODION,P: EGORIN,MJ: ENGISCH,KL: BACHUR,NR:. (1985). METABOLISM AND DISPOSITION OF MENOGARIL (NSC 269 148) IN THE RABBIT.. 45(11) |
| Amount utilized | |
| Compound isolated | |
| Disease | METABOLITE AND THEIR DISTRIBUTION AFTER ONE OR EIGHT HRS WAS N-DEMETHYL-MENOGAROL (LIVER AND KIDNEY) 7-DEOXYNOGAROL (LIVER,KIDNEY,DUODENUM,AND SMALL INTESTINE),AND N-DEMETTHYL-7-DEOXYNOGAROL (LIVER). BILIARY METABOLITES INCLUDE ALL THOSE LISTED ABOVE AND THREE UNIDENTIFIED METABOLITES. URINARY METABOLITES WERE THE SAME EXCEPT FOR 7-DEOXYNOGAROL AND N-DEMTHYLMENOGAROL. 38% OF THE DRUG WAS EXCRETED UNCHANGED IN THE URINE. |
| Dose amount | 2.5 MG |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | RABBIT |
| Per unit | KG |
| Dose expression | DOSE |