Experiment 7684
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | IV |
| Organism | Empty organism |
| Citation | CHANG,CK: WANG,YE: PAO,TY: HSU,P:. (1965). THE PHYSIOLOGIC DISPOSITION OF TETRAHYDROBERBERINE (THB).. 28() |
| Amount utilized | |
| Compound isolated | |
| Disease | 5 MINUTES AFTER ADMINISTRATION,HIGHEST CONCENTRATION IN BLOOD WAS 69 MCG/GM: WITH 10-17 MCG/GM 5-15 MINUTES LATER 70% OF DRUG BOUND TO BLOOD PROTEINS PENETRATION OF BLOOD-BRAIN BARRIER TO REACH LEVEL OF 110-180 MCG/GM IN BRAIN (2X CONCENTRATION FOUND IN BLOOD) ONE HOUR AFTER ADMINISTRATION,CONCENTRATION IN BLOOD AND BRAIN WERE MUCH LOWER THAN IN VISCERA (20 TO 50 MCG/GM). HIGHEST IN LUNG,NEXT HIGHEST IN KIDNEY,NEXT HIGHEST IN LIVER |
| Dose amount | 40.0 MG |
| Number | 2 |
| Qualitative result | ACTIVE |
| Animal | RABBIT |
| Per unit | KG |
| Dose expression | DOSE |