Experiment 776077
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | INTRAGASTRIC |
| Organism | Empty organism |
| Citation | CHEN,SJ: YANG,YM: LIU,YM: ZHANG,B: PAN,XB: ZENG,F:. (2001). PHARMACOKINETICS OF DAURICINE IN RATS.. 17(2) |
| Amount utilized | |
| Compound isolated | |
| Disease | THE PEAK PLASMA CONCN. AFTER INTRAGASTRIC (I.G.) ADMINISTRATION OF 150 MG/KG 1 WAS <1 MG/L. THE ABS. BIOAVAILABILITY WAS ABOUT 16.6%. THE PEAK TIME WAS ABOUT 15 MIN AFTER I.G. ADMINSITRATION AND INCREASED AGAIN IN 4 H. A STOMACH-INTESTINE RECIRCULATION APPEARED TO BE THE MAJOR REASON FOR THE DOUBLE PEAK PHENOMENON. DAURICINE WAS WIDELY DISTRIBUTED IN ALMOST ALL THE TISSUES AND ORGANS.FECES WERE THE MAIN ROUTE BY WHICH THE DRUG WAS EXCRETED. |
| Dose amount | 150.0 MG |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | RAT |
| Per unit | KG |
| Dose expression | DOSE |