Experiment 813478
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | IV |
| Organism | Maytenus buchananii (CELASTRACEAE) |
| Citation | BLUM,RH: KAHLERT,T:. (1978). MAYTANSINE: A PHASE I STUDY OF AN ANSA MACROLIDE WITH ANTITUMOR ACTIVITY.. 62() |
| Amount utilized | |
| Compound isolated | |
| Disease | CLINICAL TRIAL(PHASE I)IN 38 ADULT SOLID TUMOR PATIENTS FIVE DAILY BOLUS INJECTIONS WERE REPEATED AT 21 DAY INTERVALS GASTROINTESTINAL TOXICITY WAS DOSE RELATED AND DOSE LIMITING AT 0.5 MG/SQ METER OF BODY SURFACE |
| Dose amount | 0.5 MG |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | HUMAN ADULT |
| Per unit | SQ M BODY SURFACE |
| Dose expression | DOSE |
| Gender | GIVEN TO BOTH SEXES |