Experiment 815790
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | IV |
| Organism | Fusarium equiseti (HYPHOMYCETES) |
| Citation | HAAS,C: GOODWIN,W: LEITE,C: STEPHENS,R: HOOGSTRATEN,B:. (1977). PHASE I STUDY OF ANGUIDINE (DIACETYOXYSCIRPENOL NSC#1415377).. 18() |
| Amount utilized | |
| Compound isolated | |
| Disease | PHASE I CLINICAL TRIAL IN 12 PATIENTS ALL 12 HAD MODERATE TO SEVERE GI TOXICITY HYPOTENSION IN SUBJECTS AT 4.5 MG/SQ M OR ABOVE 9 PATIENTS HAD CHILLS,FEVER,AND CNS CHANGES,INCLUDING HALLUCINATIONS,CONFUSION AND ERRATIC BEHAVIOR |
| Dose amount | 6.0 MG |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | HUMAN ADULT |
| Per unit | SQ M BODY SURFACE |
| Dose expression | DOSE |