Experiment 825405
Compounds isolated
Alerts
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | IV |
| Organism | Empty organism |
| Citation | MAROUN,JA: FIELDS,AL: PATER,JL: STEWART,DJ: CRIPPS,C: EISENHAUER,E:. (1984). PHASE II STUDY OF ACIVICIN IN COLORECTAL CARCINOMA: A NATIONAL CANCER INSTITUTE OF CANADA STUDY.. 68(9) |
| Amount utilized | |
| Compound isolated | |
| Disease | IN THIS PHASE II TRIAL,20 PATIENTS WITH ADVANCED COLORECTAL CANCER WERE TREATED IN DOSES ESCALATING TO 26 MG/SQ.M IN 21 DAYS CYCLES.OF THE 17 PATIENTS EVALUABLE,THERE WAS NO OBJECTIVE RESPONSE.9 PATIENTS HAD STABLE DISEASE. HEMATOLOGICAL TOXICITY WAS MINIMAL.CNS TOXICITY WAS OBSERVED IN 11 PATIENTS CONSISTING OF CONFUSION,DEPRESSION,SLEEPING DIFFICULTY AND SENSE OF UNREALITY AND DIFFICULTY OF CONCENTRATION. |
| Dose amount | 15.0 MG |
| Number | 1 |
| Qualitative result | EQUIVOCAL |
| Animal | HUMAN ADULT |
| Per unit | SQ M BODY SURFACE |
| Dose expression | DOSE |