Experiment 838797
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | ORAL |
| Organism | Empty organism |
| Citation | GUZE,BH: BAXTER JR,LR:. (1985). BIOAVAILABILITY OF ORAL PHYSOSTIGMINE.. 313(20) |
| Amount utilized | |
| Compound isolated | |
| Disease | IN TWO PATIENTS GIVEN A SINGLE ORAL DOSE OF 1-3 MG, THE AREAS UNDER THE CURVE WAS 54 AND 17. IN ONE PATIENT GIVEN A SINGLE DOSE OF 2 MG, THE AREA UNDER THE CURVE WAS 30. HIGHEST BLOOD CONCENTRATIONS WERE COLLECTED AFTER 20 MINUTES. IN LOW DOSE PATIENTS THEY WERE 2.29 AND 0.45 NG/ML, AND 1.15 NG/ML IN THE HIGH DOSE PATIENTS. PERCENTAGE OF ORAL DOSE REACHING SYSTEMIC CIRCULATION WAS 11.7, 5.2 AND 7.8, RESP. |
| Dose amount | 1.3-2 MG |
| Number | 2 |
| Qualitative result | ACTIVE |
| Animal | HUMAN ADULT |
| Per unit | PERSON |
| Dose expression | DOSE |