Experiment 856369
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | IV INFUSION |
| Organism | Empty organism |
| Citation | LONGNECKER,SM: DONEHOWER,RC: CATES,AE: CHEN,TL: BRUNDRETT,RB: GROCHOW,LB: ETTINGER,DS: COLVIN,M:. (1987). HIGH-PERFORMANCE LIQUID CHROMATOGRAPHIC ASSAY FOR TAXOL IN HUMAN PLASMA AND URINE AND PHARMACOKINETICS IN A PHASE I TRIAL.. 71(1) |
| Amount utilized | |
| Compound isolated | |
| Disease | A PHASE 1 TRIAL. ALPHA HALF LIFE 16.2 MIN, BETA HALF LIFE 6.4 HOURS, VOLUME OF DISTRIBUTION FOR CENTRAL COMPARTMENT 8.6 L/SQ.M., AT STEADY STATE 67.1 L/SQ.M. MEAN PLASMA CLEARANCE 253 ML/MIN/SQ.M., URINARY CLEARANCE 29.3 ML/MIN/SQ.M. DOSE RANGE 15 TO 265 MG/SQ.M BY 60 TO 360 MIN INFUSION. |
| Dose amount | VAR |
| Number | 2 |
| Qualitative result | ACTIVE |
| Animal | HUMAN ADULT |
| Dose expression | DOSE |