| Disease | PARAMETERS WERE: BETA HALF LIFE,82.6 MIN,RATE CONST.,FOR TRANSFER OF DRUG FROM CENTRAL TO PERIPHERAL COMPARTMENT,0.057/MIN,RATE CONST.FOR TRANSFER FROM PERIPHERAL TO CENTRAL COMPART.,0.039/MIN:& RATE CONST.FOR ELIMINATION FROM CENTRAL COMPART.0.024/MIN
OTHER PARAMETERS WERE: VOLUME OF DISTRIBUTION (VD) OF THE CENTRAL COMPARTMENT, OF THE 2 COMPARTMENT MODEL, 70 ML/KG, VD DURING POST-DISTRIBUTIVE PHASE, 202 ML/KG,VD AT STEADY STATE, 173 ML/KG, TOTAL BODY CLEARANCE, 1.69 ML/MIN KG, AND RENAL CLEARANCE 1.03 ML/MIN KG
SIXTY ONE PERCENT WAS EXCRETED UNCHANGED IN THE URINE. |