Experiment 884491

Compounds isolated

Details

PropertyValue
Pharmacology
Administration routeINTRAGASTRIC
OrganismEmpty organism
CitationAZOULAY,P: REYNIER,JP: BALANSARD,G: GASQUET,M: TIMON-DAVID,P:. (1986). BIOGALENIC AND PHARMACOLOGICAL STUDY ON THREE SESQUITERPENES WITH ANTIPARASITIC ACTIONS: HELENIN, SANTONIN, AND 12 CARBOXY-3,11(13)-EUDESMADIENE.. 61(12)
Amount utilized
Compound isolated
DiseaseACTIVITY OF COMPOUND IN VIVO WAS POOR OWING TO CONSIDERABLE ABSORPTION IN THE DIGESTIVE TRACT, SO STANDARD GALENICAL METHODS OF ADSORPTION, MICROENCAPSULATION AND COATING WERE EVALUATED TO RETARD ABSORPTION. IMPROVEMENTS OF ABOUT 10% WERE NOTED.
Dose amountVAR
Number1
Qualitative resultACTIVE
AnimalMOUSE
Dose expressionDOSE