Experiment 917674

Details

PropertyValue
Pharmacology
Administration routeIV
OrganismEmpty organism
CitationFUJII,T: MIYAZAKI,H: NAMBU,K: KAGEMOTO,A: HASHIMOTO,M:. (1984). DISPOSITION AND METABOLISM OF 14C-DEHYDROCORYDALINE IN MICE AND RATS.. 33(8)
Amount utilized
Compound isolated
DiseaseMAXIMUM BLOOD LEVEL WAS 0.06 MCG/ML. RADIOACTIVITY WAS DISTRIBUTED IN THE GI TRACT, LIVER AND KIDNEYS. MOST ACTIVITY WAS EXCRETED IN THE FECES. EXCRETION VIA URINE AND BILE WAS MINOR. METABOLITE ANALYSIS SUGGESTED THAT THE COMPOUND WAS METABOLIZED VIA O-DEMETHYLATION AND SUBSEQUENT CONJUGATION WITH GLUCURONIC ACID.
Dose amount6.8 MG
Number4
Qualitative resultACTIVE
AnimalRAT
Per unitKG
Dose expressionDOSE