Experiment 930729

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationJENSEN,PB: SORENSEN,BS: DEMANT,EJF: SEHESTED,M: JENSEN,PS: VINDELOV,L: HANSEN,HH:. (1990). ANTAGONISTIC EFFECT OF ACLARUBICIN ON THE CYTOTOXICITY OF ETOPOSIDE AND 4'-(9-ACRIDINYLAMINO)METHANESULFON-M-ANISIDIDE IN HUMAN SMALL CELL LUNG CANCER CELL LINES AND ON TOPOISOMERASE II-MEDIATED DNA CLEAVAGE.. 50(11)
Amount utilized
Compound isolated
DiseaseINHIBITION OCCURS AT THE GIVEN CONCENTRATION AND GREATER. AT THESE CONCENTRATIONS, THE ETOPOSIDE-INDUCED FORMATION OF CLEAVABLE COMPLEXES WAS INHIBITED, WHILE CONCENTRATIONS OF 1 TO 10 NANOMOLAR HAD A SYNERGISTIC EFFECT ON SUCH FORMATION.
Dose amount1.0 MICROMOLS
Number2
Qualitative resultACTIVE
Dose expressionCONC USED