Experiment 933556
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Empty organism |
| Citation | TAKISHIMA,K: FRIEDMAN,BA: FUJIKI,H: ROSNER,MR:. (1988). THAPSIGARGIN, A NOVEL PROMOTER, PHOSPHORYLATES THE EPIDERMAL GROWTH FACTOR RECEPTOR AT THREONINE 669.. 157(2) |
| Amount utilized | |
| Compound isolated | |
| Disease | COMPOUND CAUSES PHOSPHORYLATION OF, AMONG OTHERS, THREONINE 669 OF EPIDERMAL GROWTH FACTOR RECEPTOR, A SITE NOT PHOSPHORYLATED BY PROTEIN KINASE C. THIS DECREASES AFFINITY OF RECEPTOR FOR EGF AND INHIBITS EGF-INDUCED TYROSINE KINASE ACTIVITY. |
| Dose amount | 1.0 MCG |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | CELL CULTURE |
| Per unit | ML |
| Dose expression | CONC USED |