Experiment 943827

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationZIMANYI,I: PESSAH,IN:. (1991). COMPARISON OF [3H]RYANODINE RECEPTORS AND CA++ RELEASE FROM RAT CARDIAC AND RABBIT SKELETAL MUSCLE SARCOPLASMIC RETICULUM.. 256(3)
Amount utilized
Compound isolated
DiseaseRYANODINE BINDING SITES ON SR ISOLATED FROM SKELETAL MUSCLE EXAMINED. CA++ ACTIVATES SUCH SITES. RUTHENIUM RED, MG++ & NEOMYCIN ARE POTENT INHIBITORS. BETA,GAMMA-METHYLENEADENOSINE 51-TRIPHOSPHATE ENHANCES HIGH AFFINITY BINDING(SUBOPTIMAL CA++). HIGH SALT LEVEL ENHANCES BINDING, THOUGH THE NUMBER OF BINDING SITES IS REDUCED.
Dose amountVAR
Number2
Qualitative resultACTIVE
AnimalRABBIT
Dose expressionCONC USED