Experiment 947167

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationESA,AH: BOTO,WO: ADLER,WH: MAY,WS: HESS,AD:. (1990). ACTIVATION OF T-CELLS BY BRYOSTATINS: INDUCTION OF THE IL-2 RECEPTOR GENE TRANSCRIPTION AND DOWN-MODULATION OF SURFACE RECEPTORS.. 12(5)
Amount utilized
Compound isolated
DiseaseBRYOSTATINS ARE MACROCYCLIC LACTONES ISOLATED FROM THE MARINE BRYOZOAN BUGULA NERITINA. RESULTS SHOWED THAT TREATMENT OF T CELLS WITH BRYO 1 RAPIDLY REDUCED THE SURFACE EXPRESSION OF CD4 & CD3. IN CONTRAST THE CD8 RECEPTOR WAS UNAFFECTED.
Dose amount50.0 NANOMOLS
Number2
Qualitative resultACTIVE
Dose expressionCONC USED