Experiment 947957
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Empty organism |
| Citation | RAUFMAN,JP: SINGH,L: ENG,J:. (1991). EXENDIN-3, A NOVEL PEPTIDE FROM HELODERMA HORRIDUM VENOM, INTERACTS WITH VASOACTIVE INTESTINAL PEPTIDE RECEPTORS AND A NEWLY DESCRIBED RECEPTOR ON DISPERSED ACINI FROM GUINEA PIG PANCREAS.. 266(5) |
| Amount utilized | |
| Compound isolated | |
| Disease | PANCREATIC ACINI, WHICH WERE DISPERSED AND SUSPENDED IN STANDARD INCUBATION MEDIUM, WERE ASSAYED. AN 8-FOLD INCREASE IN AMYLASE RELEASE WAS THE MAXIMAL EFFECT OBTAINED. EFFECT INHIBITED BY VIP-ANTAGONISTS. |
| Dose amount | 500.0 NANOMOLS |
| Number | 2 |
| Qualitative result | ACTIVE |
| Animal | GUINEA PIG |
| Dose expression | ED50 |