Experiment 950334
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | IV |
| Organism | Empty organism |
| Citation | SESSA,C: ZUCCHETTI,M: DAVOLI,E: CALIFANO,R: CAVALLI,F: FRUSTACI,S: GUMBRELL,L: SULKES,A: WINOGRAD,B: D'INCALCI,M:. (1991). PHASE I AND CLINICAL PHARMACOLOGICAL EVALUATION OF APHIDICOLIN GLYCINATE.. 83(16) |
| Amount utilized | |
| Compound isolated | |
| Disease | 24 PATIENTS WERE ENTERED IN A PHASE I STUDY. DAILY DOSES OF 12-2250 MG/SQ M WERE GIVEN FOR 5 DAYS EVERY 3 WEEKS. DOSE-RELATED TOXIC EFFECTS WERE PAIN ALONG VEIN OF INJECTION AND ERYTHEMA OF SURROUNDING SKIN. MILD LEUKOPENIA AND REVERSIBLE GRADE 1 INCREASE IN LIVER FUNCTION WERE ALSO OBSERVED. ANTITUMOR ACTIVITY WAS NOT OBSERVED. |
| Dose amount | VAR |
| Number | 1 |
| Qualitative result | . |
| Animal | HUMAN ADULT |
| Dose expression | DOSE |