Experiment 950404
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Boerhavia diffusa (NYCTAGINACEAE) |
| Citation | LAMI,N: KADOTA,S: KIKUCHI,T: MOMOSE,Y:. (1991). CONSTITUENTS OF THE ROOTS OF BOERHAAVIA DIFFUSA L. III. IDENTIFICATION OF CA2 CHANNEL ANTAGONISTIC COMPOUND FROM THE METHANOL EXTRACT.. 39(6) |
| Amount utilized | |
| Compound isolated | |
| Disease | IN FROG ATRIAL CELLS, AN ACTION POTENTIAL CAN BE TRIGGERED EVEN AFTER TRANSIENT NA+ CURRENT HAS BEEN BLOCKED BY TETRODOTOXIN. THE PEAK HEIGHT AND DURATION OF THIS SLOW RESPONSE ARE MODULATED BY CA++ CURRENT. THE GIVEN COMPOUND DECREASES HEIGHT AND INCREASES DURATION BY BLOCKING THIS CA++ CURRENT. |
| Dose amount | 10.0 MILLIMOLS |
| Number | 2 |
| Qualitative result | ACTIVE |
| Animal | CELL CULTURE |
| Dose expression | CONC USED |