Experiment 952345

Details

PropertyValue
Pharmacology
OrganismMollisia ventosa (DERMATEACEAE)
CitationNAKANISHI,S: KURODA,K: OSAWA,K: KASE,H:. (1990). CALMODULIN ANTAGONISTIC ACTION OF KS-504A, A NOVEL METABOLITE OF THE FUNGUS MOLLISIA VENTOSA.. 54(10)
Amount utilized
Compound isolated
DiseaseCOMPOUND INTERACTS WITH CALMODULIN TO INHIBIT MYOSIN LIGHT CHAIN KINASE. THIS EFFECT WAS COMPETITIVE WITH RESPECT TO CALMODULIN AND NON-COMPETITIVE WITH RESPECT TO ATP.
Dose amount6.3 MICROMOLS
Number4
Qualitative resultACTIVE
Dose expressionIC50