Experiment 952430
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Empty organism |
| Citation | SCHONTHAL,A: SUGARMAN,J: BROWN,JH: HANLEY,MR: FERAMISCO,JR:. (1991). REGULATION OF C-FOS AND C-JUN PROTOONCOGENE EXPRESSION BY THE CA2+-ATPASE INHIBITOR THAPSIGARGIN.. 88(16) |
| Amount utilized | |
| Compound isolated | |
| Disease | COMPOUND INDUCED EXPRESSION OF PROTO-ONCOGENES C-FOS + C-JUN SHOWN BY ACCUMULATION OF RELATED M-RNA. COADMINISTRATION OF TPA HAD A SYNERGISTIC EFFECT ON C-FOS EXPRESSION ONLY. COMPOUND HAD NO EFFECT ON BASAL OR PHORBOL ESTER-INDUCED PROTEIN KINASE C ACTIVITY. INHIBITION OR DEPLETION OF PKC PARTIALLY DIMINISHED THE C-FOS BUT NOT THE C-JUN RESPONSE. |
| Dose amount | 100.0 NANOMOLS |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | CELL CULTURE |
| Dose expression | CONC USED |